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1

Melanocortin Receptors: Identification and Characterization by Melanotropic Peptide Agonists and Antagonists

MAC E. HADLEY, VICTOR J. HRUBY, JIWEN JIANG, SHUBH D. SHARMA, JODY L. FINK, CARRIE HASKELL-LUEVANO, DAVID L. BENTLEY, FAHAD AL-OBEIDI, TOMI K. SAWYER

Journal:

Pigment Cell & Melanoma Research

Year:

1996

Language:

english

File:

PDF, 2.51 MB

english, 1996

2

The 1,4-Benzodiazepine-2,5-dione Small Molecule Template Results in Melanocortin Receptor Agonists with Nanomolar Potencies

Joseph, Christine G., Wilson, Krista R., Wood, Michael S., Sorenson, Nicholas B., Phan, Dong V., Xiang, Zhimin, Witek, Rachel M., Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 297 KB

english, 2008

3

α-MSH tripeptide analogs activate the melanocortin 1 receptor and reduce UV-induced DNA damage in human melanocytes

Zalfa A. Abdel-Malek, Andrew Ruwe, Renny Kavanagh-Starner, Ana Luisa Kadekaro, Viki Swope, Carrie Haskell-Luevano, Leonid Koikov, James J. Knittel

Journal:

Pigment Cell & Melanoma Research

Year:

2009

Language:

english

File:

PDF, 365 KB

english, 2009

4

Discovery of Prototype Peptidomimetic Agonists at the Human Melanocortin Receptors MC1R and MC4R

Haskell-Luevano, Carrie, Hendrata, Siska, North, Cheryl, Sawyer, Tomi K., Hadley, Mac E., Hruby, Victor J., Dickinson, Chris, Gantz, Ira

Journal:

Journal of Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 214 KB

english, 1997

5

Biological and Conformational Examination of Stereochemical Modifications Using the Template Melanotropin Peptide, Ac-Nle-c[Asp-His-Phe-Arg-Trp- Ala-Lys]-NH 2 , on Human Melanocortin Receptors

Haskell-Luevano, Carrie, Nikiforovich, Gregory, Sharma, Shubh D., Yang, Ying-Kui, Dickinson, Chris, Hruby, Victor J., Gantz, Ira

Journal:

Journal of Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 332 KB

english, 1997

6

Structure-Activity Relationship Studies of a Macrocyclic AGRP-Mimetic Scaffold c[Pro-Arg-Phe-Phe-Asn-Ala-Phe-DPro] Yield Potent and Selective Melanocortin-4 Receptor Antagonists and Melanocortin-5 Receptor Inverse Agonists that Increase Food Intake in Mice

Fleming, Katlyn A., Ericson, Mark D., Freeman, Katie T., Adank, Danielle N., Lunzer, Mary M., Wilber, Stacey L, Haskell-Luevano, Carrie

Journal:

ACS Chemical Neuroscience

Year:

2018

Language:

english

File:

PDF, 1.08 MB

english, 2018

7

Allosteric Modulators of Drug Targets Special Issue

Haskell-Luevano, Carrie, Georg, Gunda I., Wang, Shaomeng, Meanwell, Nicholas

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 253 KB

english, 2018

8

Design of peptides, proteins, and peptidomimetics in chi space

Victor J. Hruby, Guigen Li, Carrie Haskell-Luevano, Mark Shenderovich

Journal:

Year:

1997

Language:

english

File:

PDF, 1.29 MB

english, 1997

9

Structure-activity relationship and metabolic stability studies of backbone cyclization and N-methylation of melanocortin peptides

Yaniv Linde, Oded Ovadia, Eli Safrai, Zhimin Xiang, Federico P. Portillo, Deborah E. Shalev, Carrie Haskell-Luevano, Amnon Hoffman, Chaim Gilon

Journal:

Year:

2008

Language:

english

File:

PDF, 314 KB

english, 2008

10

Melanocortin Ligands: 30 Years of Structure—Activity Relationship (SAR) Studies

Jerry Ryan Holder, Carrie Haskell-Luevano

Journal:

Year:

2004

File:

PDF, 51 KB

2004

11

Current Trends in the Structure—Activity Relationship Studies of the Endogenous Agouti-Related Protein (AGRP) Melanocortin Receptor Antagonist

Andrzej M. Wilczynski, Christine G. Joseph, Carrie Haskell-Luevano

Journal:

Year:

2005

File:

PDF, 8 KB

2005

12

Melanocortin ligands: 30 years of structure–activity relationship (SAR) studies

Jerry Ryan Holder, Carrie Haskell-Luevano

Journal:

Medicinal Research Reviews

Year:

2004

Language:

english

File:

PDF, 391 KB

english, 2004

13

Current trends in the structure—activity relationship studies of the endogenous agouti-related protein (AGRP) melanocortin receptor antagonist

Andrzej M. Wilczynski, Christine G. Joseph, Carrie Haskell-Luevano

Journal:

Medicinal Research Reviews

Year:

2005

Language:

english

File:

PDF, 264 KB

english, 2005

14

β-Turn secondary structure and melanocortin ligands

Erica M. Haslach, Jay W. Schaub, Carrie Haskell-Luevano

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 574 KB

english, 2009

15

The effect of backbone cyclization on PK/PD properties of bioactive peptide-peptoid hybrids: The melanocortin agonist paradigm

Oded Ovadia, Yaniv Linde, Carrie Haskell-Luevano, Marvin L. Dirain, Tanya Sheynis, Raz Jelinek, Chaim Gilon, Amnon Hoffman

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 496 KB

english, 2010

16

Design and pharmacology of peptoids and peptide–peptoid hybrids based on the melanocortin agonists core tetrapeptide sequence

Jerry Ryan Holder, Rayna M Bauzo, Zhimin Xiang, Joseph Scott, Carrie Haskell-Luevano

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 205 KB

english, 2003

17

Semi-rigid tripeptide agonists of melanocortin receptors

Andrew R. Ruwe, Leonid Koikov, Zalfa Abdel-Malek, Carrie Haskell-Luevano, Marvin L. Dirain, Federico Portillo, Zhimin Xiang, Matt Wortman, James J. Knittel

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 658 KB

english, 2009

18

Urea small molecule agonists on mouse melanocortin receptors

Christine G. Joseph, Rayna M. Bauzo, Zhimin Xiang, Carrie Haskell-Luevano

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 171 KB

english, 2003

19

Facile removal of theN-indole-mesitylenesulfonyl protecting group using HF cleavage conditions

Carrie Haskell-Luevano, Lakmal W. Boteju, Victor J. Hruby

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1995

Language:

english

File:

PDF, 496 KB

english, 1995

20

Molecular Mechanism of the Constitutive Activation of the L250Q Human Melanocortin-4 Receptor Polymorphism

Bettina Proneth, Zhimin Xiang, Irina D. Pogozheva, Sally A. Litherland, Oleg S. Gorbatyuk, Amanda M. Shaw, William J. Millard, Henry I. Mosberg, Carrie Haskell-Luevano

Journal:

Chemical Biology & Drug Design

Year:

2006

Language:

english

File:

PDF, 959 KB

english, 2006

21

Structure–Activity Relationships of Melanocortin Agonists Containing the Benzimidazole Scaffold

Aleksandar Todorovic, Christine G. Joseph, Nicholas B. Sorensen, Michael S. Wood, Carrie Haskell-Luevano

Journal:

Chemical Biology & Drug Design

Year:

2007

Language:

english

File:

PDF, 624 KB

english, 2007

22

Microwave-Assisted Solid-Phase Peptide Synthesis Utilizing N-Fmoc-Protected (α-aminoacyl)benzotriazoles

Alan R. Katritzky, Niveen M. Khashab, Megumi Yoshioka, Danniebelle N. Haase, Krista R. Wilson, Jodie V. Johnson, Alfred Chung, Carrie Haskell-Luevano

Journal:

Chemical Biology & Drug Design

Year:

2007

Language:

english

File:

PDF, 107 KB

english, 2007

23

The Proopiomelanocortin System

MAC E. HADLEY, CARRIE HASKELL-LUEVANO

Journal:

Annals of the New York Academy of Sciences

Year:

1999

Language:

english

File:

PDF, 951 KB

english, 1999

24

Melanocortin Tetrapeptides Modified at the N-Terminus, His, Phe, Arg, and Trp Positions

JERRY RYAN HOLDER, CARRIE HASKELL-LUEVANO

Journal:

Annals of the New York Academy of Sciences

Year:

2003

File:

PDF, 4.67 MB

2003

25

Use of chimeric melanocortin-2 and -4 receptors to identify regions responsible for ligand specificity and dependence on melanocortin 2 receptor accessory protein

Patricia M. Hinkle, Madhavika N. Serasinghe, Andrea Jakabowski, Julien A. Sebag, Krista R. Wilson, Carrie Haskell-Luevano

Journal:

European Journal of Pharmacology

Year:

2011

Language:

english

File:

PDF, 1.34 MB

english, 2011

26

Effect of serotonergic anorectics on food intake and induction of Fos in brain of mice with disruption of melanocortin 3 and/or 4 receptors

Neil E. Rowland, Kaihan J. Fakhar, Kimberly L. Robertson, Carrie Haskell-Luevano

Journal:

Pharmacology Biochemistry and Behavior

Year:

2010

Language:

english

File:

PDF, 330 KB

english, 2010

27

Characterization of aliphatic, cyclic, and aromatic N-terminally “capped” His-d-Phe-Arg-Trp-NH2 tetrapeptides at the melanocortin receptors

Jerry Ryan Holder, Fernanda F Marques, Zhimin Xiang, Rayna M Bauzo, Carrie Haskell-Luevano

Journal:

European Journal of Pharmacology

Year:

2003

Language:

english

File:

PDF, 590 KB

english, 2003

28

Chimeric NDP-MSH and MTII melanocortin peptides with agouti-related protein (AGRP) Arg-Phe-Phe amino acids possess agonist melanocortin receptor activity

Christine G. Joseph, Andrzej Wilczynski, Jerry R. Holder, Zhimin Xiang, Rayna M. Bauzo, Joseph W. Scott, Carrie Haskell-Luevano

Journal:

Year:

2003

Language:

english

File:

PDF, 149 KB

english, 2003

29

Feeding effects of melanocortin ligands—A historical perspective

Boman G. Irani, Carrie Haskell-Luevano

Journal:

Year:

2005

Language:

english

File:

PDF, 227 KB

english, 2005

30

A review of melanocortin receptor small molecule ligands

Aleksandar Todorovic, Carrie Haskell-Luevano

Journal:

Year:

2005

Language:

english

File:

PDF, 238 KB

english, 2005

31

Ghrelin-induced food intake and growth hormone secretion are altered in melanocortin 3 and 4 receptor knockout mice

Amanda M. Shaw, Boman G. Irani, Marcus C. Moore, Carrie Haskell-Luevano, William J. Millard

Journal:

Year:

2005

Language:

english

File:

PDF, 167 KB

english, 2005

32

Melanocortin-4 receptor-null mice display normal affective licking responses to prototypical taste stimuli in a brief-access test

Shachar Eylam, Marcus Moore, Carrie Haskell-Luevano, Alan C. Spector

Journal:

Year:

2005

Language:

english

File:

PDF, 249 KB

english, 2005

33

Physiology and chemistry of the melanocortin pathway

Carrie Haskell-Luevano

Journal:

Year:

2006

Language:

english

File:

PDF, 74 KB

english, 2006

34

Functional characterization of the modified melanocortin peptides responsible for ligand selectivity at the human melanocortin receptors

Min Chen, Keith E. Georgeson, Carroll M. Harmon, Carrie Haskell-Luevano, Yingkui Yang

Journal:

Year:

2006

Language:

english

File:

PDF, 910 KB

english, 2006

35

γ2-Melanocyte stimulation hormone (γ2-MSH) truncation studies results in the cautionary note that γ2-MSH is not selective for the mouse MC3R over the mouse MC5R

Christine G. Joseph, Hua Yao, Joseph W. Scott, Nicholas B. Sorensen, Rebecca N. Marnane, Kathleen G. Mountjoy, Carrie Haskell-Luevano

Journal:

Year:

2010

Language:

english

File:

PDF, 532 KB

english, 2010

36

Effect of MTII on food intake and brain c-Fos in melanocortin-3, melanocortin-4, and double MC3 and MC4 receptor knockout mice

Neil E. Rowland, Jay W. Schaub, Kimberly L. Robertson, Amy Andreasen, Carrie Haskell-Luevano

Journal:

Year:

2010

Language:

english

File:

PDF, 230 KB

english, 2010

37

Agouti-related protein functions as an inverse agonist at a constitutively active brain melanocortin-4 receptor

Carrie Haskell-Luevano, Eileen K Monck

Journal:

Regulatory Peptides

Year:

2001

Language:

english

File:

PDF, 248 KB

english, 2001

38

The agouti-related protein decapeptide (Yc[CRFFNAFC]Y) possesses agonist activity at the murine melanocortin-1 receptor

Carrie Haskell–Luevano, Eileen K Monck, Y.-P Wan, Anzeela M Schentrup

Journal:

Year:

2000

Language:

english

File:

PDF, 181 KB

english, 2000

39

Elongation studies of the human agouti-related protein (AGRP) core decapeptide (Yc[CRFFNAFC]Y) results in antagonism at the mouse melanocortin-3 receptor

Christine G Joseph, Rayna M Bauzo, Zhimin Xiang, Amanda M Shaw, William J Millard, Carrie Haskell-Luevano

Journal:

Year:

2003

Language:

english

File:

PDF, 103 KB

english, 2003

40

Structure–activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the mouse melanocortin receptors: Part 3: modifications at the Arg position

Jerry Ryan Holder, Zhimin Xiang, Rayna M Bauzo, Carrie Haskell-Luevano

Journal:

Year:

2003

Language:

english

File:

PDF, 284 KB

english, 2003

41

Structure activity studies of the melanocortin antagonist SHU9119 modified at the 6, 7, 8, and 9 positions☆

Carrie Haskell–Luevano, Sejin Lim, Wei Yuan, Roger D Cone, Victor J Hruby

Journal:

Year:

2000

Language:

english

File:

PDF, 146 KB

english, 2000

42

Structure–Activity Relationships of Peptides Incorporating a Bioactive Reverse-Turn Heterocycle at the Melanocortin Receptors: Identification of a 5800-fold Mouse Melanocortin-3 Receptor (mMC3R) Selective Antagonist/Partial Agonist versus the Mouse Melanocortin-4 Receptor (mMC4R)

Singh, Anamika, Dirain, Marvin, Witek, Rachel, Rocca, James R., Edison, Arthur S., Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 3.78 MB

english, 2013

43

A Solid-Phase Approach to Mouse Melanocortin Receptor Agonists Derived from a Novel Thioether Cyclized Peptidomimetic Scaffold

Bondebjerg, Jon, Xiang, Zhimin, Bauzo, Rayna M., Haskell-Luevano, Carrie, Meldal, Morten

Journal:

Journal of the American Chemical Society

Year:

2002

Language:

english

File:

PDF, 199 KB

english, 2002

44

Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH 2 at the Mouse Melanocortin Receptors: Part 2 Modifications at the Phe Position

Holder, Jerry Ryan, Bauzo, Rayna M., Xiang, Zhimin, Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 104 KB

english, 2002

45

N-Terminal Fatty Acylated His- d Phe-Arg-Trp-NH 2 Tetrapeptides: Influence of Fatty Acid Chain Length on Potency and Selectivity at the Mouse Melanocortin Receptors and Human Melanocytes

Todorovic, Aleksandar, Holder, Jerry Ryan, Bauzo, Rayna M., Scott, Joseph Walker, Kavanagh, Renny, Abdel-Malek, Zalfa, Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 234 KB

english, 2005

46

Incorporation of a Bioactive Reverse-Turn Heterocycle into a Peptide Template Using Solid-Phase Synthesis To Probe Melanocortin Receptor Selectivity and Ligand Conformations by 2D 1 H NMR

Singh, Anamika, Wilczynski, Andrzej, Holder, Jerry R., Witek, Rachel M., Dirain, Marvin L., Xiang, Zhimin, Edison, Arthur S., Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 3.34 MB

english, 2011

47

Compounds That Activate the Mouse Melanocortin-1 Receptor Identified by Screening a Small Molecule Library Based upon the β-Turn

Haskell-Luevano, Carrie, Rosenquist, Åsa, Souers, Andrew, Khong, Kathy C., Ellman, Jonathon A., Cone, Roger D.

Journal:

Journal of Medicinal Chemistry

Year:

1999

Language:

english

File:

PDF, 187 KB

english, 1999

48

Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His- d -Phe-Arg-Trp-NH 2 at the Mouse Melanocortin Receptors. 4. Modifications at the Trp Position

Holder, Jerry Ryan, Xiang, Zhimin, Bauzo, Rayna M., Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 149 KB

english, 2002

49

Pharmacological Characterization of 40 Human Melanocortin-4 Receptor Polymorphisms with the Endogenous Proopiomelanocortin-Derived Agonists and the Agouti-Related Protein (AGRP) Antagonist †,‡

Xiang, Zhimin, Litherland, Sally A., Sorensen, Nicholas B., Proneth, Bettina, Wood, Michael S., Shaw, Amanda M., Millard, William J., Haskell-Luevano, Carrie

Journal:

Year:

2006

Language:

english

File:

PDF, 328 KB

english, 2006

50

Structural Characterization and Pharmacology of a Potent (Cys101−Cys119, Cys110−Cys117) Bicyclic Agouti-Related Protein (AGRP) Melanocortin Receptor Antagonist

Wilczynski, Andrzej, Wang, Xiang S., Bauzo, Rayna M., Xiang, Zhimin, Shaw, Amanda M., Millard, William J., Richards, Nigel G., Edison, Arthur S., Haskell-Luevano, Carrie

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 438 KB

english, 2004

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